天衡药研长期为国内外客户提供多种高品质医药中间体,4500㎡化工车间软硬件齐全,可以实现的反应类型包括不对称合成、高压氢化、空气和水敏感反应、金属催化、氧化还原反应等。
— 目前可提供中间体 —
产品名称 Product name |
登记号 CAS No. |
标准 Standard |
结构式 Structueal Formula |
|
伏格列波糖及中间体Voglibose & Intermediates |
伏格列波糖Voglibose |
83480-29-9 |
JP16IP In house |
|
2,3,4,6-四-O-苄基-α-D-葡萄糖 2,3,4,6-Tetra-O-benzyl-α-D-glucopyranose |
4132-28-9 6564-72-3 |
≥99% In house |
|
|
(2R,3S,4S,5S)-5-羟基-2,3,4-三(苄氧基)-5-[(苄氧基)甲基]-环己酮 (2R,3S,4S,5S)-5-Hydroxy-2,3,4-tris(phenylmethoxy)-5-[(phenylmethoxy)methyl]-cyclohexanone |
115250-38-9 |
≥99% In house |
|
|
四苄基伏格列波糖Tetra-Benzyl-Voglibose |
115250-39-0 |
≥99% In house |
|
|
盐酸厄洛替尼中间体Erlotinib Hydrochloride Intermediate |
6,7-双(甲氧基乙氧基)喹唑啉酮 6,7-Bis-(2-methoxyethoxy)-4(3H)-quinazolinone |
179688-29-0 |
≥99% In house |
|
帕利哌酮及中间体Paliperidone & Intermediates |
帕利哌酮Paliperidone |
144598-75-4 |
≥99% In house |
|
帕利哌酮棕榈酸酯Paliperidone Palmitate |
199739-10-1 |
≥99% In house |
|
|
3-(2-氯乙基)-6,7,8,9-四氢-9-羟基-2-甲基-4H-吡啶并[1,2-a]嘧啶-4-酮 3-(2-Chloroethyl)-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one |
130049-82-0 |
≥99% In house |
|
|
6-氟-3-哌啶-4-基-1,2-苯并异噁唑盐酸盐 6-Fluoro-3-(4-piperidinyl)-1,2-benzisoxazole hydrochloride |
84163-13-3 |
≥99% In house |
|
|
阿加曲班中间体Argatroban Intermediate |
(2R,4R)-4-甲基-2-哌啶甲酸乙酯Ethyl (2R,4R)-4-methyl-2-piperidinecarboxylate |
74892-82-3 |
≥99% In house |
|
盐酸吉西他滨中间体Gemcitabine Hydrochloride Intermediate |
2-脱氧-2,2二氟-戊呋喃糖-1-酮-3,5-二苯甲酸酯(T6) 2-Deoxy-2,2-difluoro-D-erythro-pentafuranous-1-ulose-3,5-dibenzoate |
122111-01-7 |
≥99% In house |
|
帕布昔利布中间体Palbociclib Intermediates |
4-(6-氨基吡啶-3-基)哌嗪-1-羧酸叔丁酯 4-(6-Aminopyridin-3-yl)piperazine-1-carboxylic acid tert-butyl este |
571188-59-5 |
≥99% In house |
|
6-溴-2-氯-8-环戊基-5-甲基-吡啶并[2,3-D]嘧啶-7(8H)-酮 6-bromo-2-chloro-8-cyclopentyl-5-Methylpyrido[2,3-d]pyriMidin-7(8H)-one |
1016636-76-2 |
≥99% In house |
|
|
奥格列汀中间体OmarigliptinIntermediates |
(2R,3S,5R)-2-(2,5-二氟苯基)-5-[2-(甲基磺酰基)-2,6-二氢吡咯并[3,4-c]吡唑-5(4H)-基]四氢-2H-吡喃-3-胺 (2R,3S,5R)-2-(2,5-Difluorophenyl)-5-[2-(methylsulfonyl)-2,6-dihydropyrrolo[3,4-c]pyrazol-5(4H)-yl]tetrahydro-2H-pyran-3-amine |
1226781-44-7 |
≥99% In house |
|
N-[(2R,3S)-2-(2,5-二氟苯基)四氢-5-氧代-2H-吡喃-3-基]氨基甲酸叔丁酯 N-[(2R,3S)-2-(2,5-Difluorophenyl)tetrahydro-5-oxo-2H-pyran-3-yl]carbamicacid1,1-dimethylethylester |
951127-25-6 |
≥99% In house |
|
|
2-(甲基磺酰)-2,4,5,6-四氢吡咯并[3,4-c]吡唑苯磺酸盐 2,4,5,6-Tetrahydro-2-(methylsulfonyl)pyrrolo[3,4-c]pyrazole benzenesulfonate |
1280210-80-1 |
≥99% In house |
|