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中间体


天衡药研长期为国内外客户提供多种高品质医药中间体,4500㎡化工车间软硬件齐全,可以实现的反应类型包括不对称合成、高压氢化、空气和水敏感反应、金属催化、氧化还原反应等。

 

产品名称
Product name

登记号
CAS No.

标准
Standard

结构式
Structueal Formula

伏格列波糖及中间体

Voglibose & Intermediates

伏格列波糖Voglibose

83480-29-9

JP16IP
In house

2,3,4,6-四-O-苄基-α-D-葡萄糖
2,3,4,6-Tetra-O-benzyl-α-D-glucopyranose

4132-28-9
6564-72-3

≥99%
In house

(2R,3S,4S,5S)-5-羟基-2,3,4-三(苄氧基)-5-[(苄氧基)甲基]-环己酮
(2R,3S,4S,5S)-5-Hydroxy-2,3,4-tris(phenylmethoxy)-5-[(phenylmethoxy)methyl]-cyclohexanone

115250-38-9

≥99%
In house

四苄基伏格列波糖Tetra-Benzyl-Voglibose

115250-39-0

≥99%
In house

盐酸厄洛替尼中间体

Erlotinib Hydrochloride Intermediate

6,7-双(甲氧基乙氧基)喹唑啉酮
6,7-Bis-(2-methoxyethoxy)-4(3H)-quinazolinone

179688-29-0

≥99%
In house

帕利哌酮及中间体

Paliperidone & Intermediates

帕利哌酮Paliperidone

144598-75-4

≥99%
In house

帕利哌酮棕榈酸酯Paliperidone Palmitate

199739-10-1

≥99%
In house

3-(2-氯乙基)-6,7,8,9-四氢-9-羟基-2-甲基-4H-吡啶并[1,2-a]嘧啶-4-酮
3-(2-Chloroethyl)-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one

130049-82-0

≥99%
In house

6-氟-3-哌啶-4-基-1,2-苯并异噁唑盐酸盐
6-Fluoro-3-(4-piperidinyl)-1,2-benzisoxazole hydrochloride

84163-13-3

≥99%
In house

阿加曲班中间体

Argatroban Intermediate

(2R,4R)-4-甲基-2-哌啶甲酸乙酯Ethyl
(2R,4R)-4-methyl-2-piperidinecarboxylate

74892-82-3

≥99%
In house

盐酸吉西他滨中间体

Gemcitabine Hydrochloride Intermediate

2-脱氧-2,2二氟-戊呋喃糖-1-酮-3,5-二苯甲酸酯(T6)
2-Deoxy-2,2-difluoro-D-erythro-pentafuranous-1-ulose-3,5-dibenzoate

122111-01-7

≥99%
In house

帕布昔利布中间体

Palbociclib Intermediates

4-(6-氨基吡啶-3-基)哌嗪-1-羧酸叔丁酯
4-(6-Aminopyridin-3-yl)piperazine-1-carboxylic acid tert-butyl este

571188-59-5

≥99%
In house

 

6-溴-2-氯-8-环戊基-5-甲基-吡啶并[2,3-D]嘧啶-7(8H)-酮
6-bromo-2-chloro-8-cyclopentyl-5-Methylpyrido[2,3-d]pyriMidin-7(8H)-one

1016636-76-2

≥99%
In house

奥格列汀中间体

OmarigliptinIntermediates

(2R,3S,5R)-2-(2,5-二氟苯基)-5-[2-(甲基磺酰基)-2,6-二氢吡咯并[3,4-c]吡唑-5(4H)-基]四氢-2H-吡喃-3-胺
(2R,3S,5R)-2-(2,5-Difluorophenyl)-5-[2-(methylsulfonyl)-2,6-dihydropyrrolo[3,4-c]pyrazol-5(4H)-yl]tetrahydro-2H-pyran-3-amine

1226781-44-7

≥99%
In house

N-[(2R,3S)-2-(2,5-二氟苯基)四氢-5-氧代-2H-吡喃-3-基]氨基甲酸叔丁酯
N-[(2R,3S)-2-(2,5-Difluorophenyl)tetrahydro-5-oxo-2H-pyran-3-yl]carbamicacid1,1-dimethylethylester

951127-25-6

≥99%
In house

2-(甲基磺酰)-2,4,5,6-四氢吡咯并[3,4-c]吡唑苯磺酸盐
2,4,5,6-Tetrahydro-2-(methylsulfonyl)pyrrolo[3,4-c]pyrazole benzenesulfonate

1280210-80-1

≥99%
In house